Sibiriline, a new small chemical inhibitor of receptor-interacting protein kinase 1, prevents immune-dependent hepatitis
F. Le Cann
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C. Delehouzé
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S. Leverrier-Penna
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A. Filliol
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A. Comte
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hal-01616420v1
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Microwave synthesis of new 3-(3-aminopropyl)-5-arylidene-2-thioxo-1,3-thiazolidine-4-ones as potential Ser/Thr protein kinase inhibitors
Camille Déliko Dago
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Wacothon Karime Coulibaly
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Yves-Alain Bekro
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Janat A. Mamyrbekova-Bekro
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Beatrice Foll-Josselin
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hal-01414293v1
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Synthesis of N-pyridyl azoles using a deprotometalation-iodolysis-N-arylation sequence and evaluation of their antiproliferative activity in melanoma cells
Madani Hedidi
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Julien Maillard
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William Erb
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Frédéric Lassagne
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Yury Halauko
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hal-03875302v1
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Development of new highly potent imidazo[1,2-b]pyridazines targeting Toxoplasma gondii calcium-dependent protein kinase 1
Espérance Moine
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Isabelle Dimier-Poisson
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Cécile Enguehard-Gueiffier
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Cédric Logé
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Mélanie Pénichon
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et al.
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hal-02389861v1
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Further investigation of Paprotrain: Towards the conception of selective and multi-targeted CNS kinase inhibitors
Christophe Labrière
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Olivier Lozach
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Mélina Blairvacq
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Laurent Meijer
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Catherine Guillou
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hal-01517780v1
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Développement de nouveaux inhibiteurs de TgCDPK1 à visée anti-toxoplasmique
Espérance Moine
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Isabelle Dimier-Poisson
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Cécile Enguehard-Gueiffier
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Cedric Logé
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Mélanie Pénichon
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6. Journées du Consortium antiParasitaire et antiFongique : CaPF-2016 " A la croisée des Mondes !" , Consortium Anti-Parasitaire et Fongique (CaPF). FRA., Mar 2016, Tours, France. 49 p
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hal-02739722v1
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From Peptide Aptamers to Inhibitors of FUR, Bacterial Transcriptional Regulator of Iron Homeostasis and Virulence
Sophie Mathieu
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Cheickna Cissé
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Sylvie Vitale
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Aynur Ahmadova
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Mélissa Degardin
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et al.
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hal-01354302v1
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Novel optimization of valmerins (tetrahydropyrido[1,2-a]isoindolones) as potent dual CDK5/GSK3 inhibitors
Aziz Ouach
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Rajâa Boulahjar
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Christine Vala
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Stéphane Bourg
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Pascal Bonnet
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et al.
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hal-01295635v1
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Synthesis, antileishmanial activity and cytotoxicity of 2,3-diaryl- and 2,3,8-trisubstituted imidazo[1,2-a]pyrazines
Pascal Marchand
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Marc-Antoine Bazin
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Fabrice Pagniez
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Guillaume Rivière
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Lizeth Bodero
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hal-03216056v1
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New insight in ARX-mutated patients' language specific impairment and underlying FOXP1 dysregulation
A. Curie
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G. Friocourt
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S. Bertrand
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F. Rochefort
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N. Loaëc
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et al.
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hal-02871228v1
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Synthesis and molecular modelling studies of 8-arylpyrido[3',2':4,5thieno[3,2-d]pyrimidin-4-amines as multitarget Ser/Thr kinases inhibitors
Yvonnick Loidreau
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Emmanuel Deau
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Pascal Marchand
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Marie-Renée Nourrisson
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Cédric Logé
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et al.
Journal articles
hal-01135195v1
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The pathogenic m.8993 T > G mutation in mitochondrial ATP6 gene prevents proton release from the subunit c -ring rotor of ATP synthase
Xin Su
,
Alain Dautant
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Malgorzata Rak
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François Godard
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Nahia Ezkurdia
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et al.
Journal articles
hal-03830051v1
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Deregulating mitochondrial metabolite and ion transport has beneficial effects in yeast and human cellular models for NARP syndrome
Xin Su
,
Malgorzata Rak
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Emmanuel Tetaud
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François Godard
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Elodie Sardin
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et al.
Journal articles
hal-02362008v1
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Tampering with Cell Division by Using Small-Molecule Inhibitors of CDK-CKS Protein Interactions
Amel Hamdi
,
Aurélien Lesnard
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Peggy Suzanne
,
Thomas Robert
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Maria A. Miteva
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et al.
Journal articles
istex
hal-02043908v1
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