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Synthetic Development of New 3-(4-Arylmethylamino)butyl-5-arylidene-rhodanines under Microwave Irradiation and Their Effects on Tumor Cell Lines and against Protein Kinases

Camille Déliko Dago , Christelle Ambeu , Wacothon-Karime Coulibaly , Yves-Alain Békro , Janat Mamyrbékova , et al.
Molecules, 2015, 20 (7), pp.12412-12435. ⟨10.3390/molecules200712412⟩
Journal articles hal-01187427v1
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Marine-Derived 2-Aminoimidazolone Alkaloids. Leucettamine B-Related Polyandrocarpamines Inhibit Mammalian and Protozoan DYRK & CLK Kinases

Nadège Loaëc , Eletta Attanasio , Benoît Villiers , Emilie Durieu , Tania Tahtouh , et al.
Marine drugs, 2017, 15 (10), pp.316 -. ⟨10.3390/md15100316⟩
Journal articles hal-01640115v1
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From Quinoxaline, Pyrido[2,3-b]pyrazine and Pyrido[3,4-b]pyrazine to Pyrazino-Fused Carbazoles and Carbolines

Frédéric Lassagne , Timothy Langlais , Elsa Caytan , Emmanuelle Limanton , Ludovic Paquin , et al.
Molecules, 2018, 23 (11), pp.2961. ⟨10.3390/molecules23112961⟩
Journal articles hal-03867783v1
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Synthesis of N-pyridyl azoles using a deprotometalation-iodolysis-N-arylation sequence and evaluation of their antiproliferative activity in melanoma cells

M. Hedidi , W. Erb , G. Bentabed-Ababsa , Floris Chevallier , L. Picot , et al.
Tetrahedron, 2016, 72 (41), pp.6467--6476. ⟨10.1016/j.tet.2016.08.056⟩
Journal articles hal-01381138v1
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High-Throughput Screening of marine resources

Arnaud Hochard , Luc Reininger , Sandrine Ruchaud , Stéphane Bach
Outstanding Marine Molecules, 2015, ⟨10.1002/9783527681501.ch23⟩
Book sections hal-03871307v1
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Redescription and phylogenetic analyses of Durchoniella spp. (Ciliophora, Astomatida) associated with the polychaete Cirriformia tentaculata (Montagu, 1808)

Laure Sauvadet , Denis H. Lynn , Erwan Roussel , Sophie Le Panse , Estelle Bigeard , et al.
European Journal of Protistology, 2017, 61 (Part A), pp.265-277. ⟨10.1016/j.ejop.2017.06.007⟩
Journal articles hal-01578167v1
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Structure-based design of novel quinoxaline-2-carboxylic acids and analogues as Pim-1 inhibitors

Bruno Oyallon , Marie Brachet-Botineau , Cédric Logé , Pascal Bonnet , Mohamed Souab , et al.
European Journal of Medicinal Chemistry, 2018, 154, pp.101-109. ⟨10.1016/j.ejmech.2018.04.056⟩
Journal articles hal-03408667v1
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The Anti-Candida albicans Agent 4-AN Inhibits Multiple Protein Kinases

Maciej Masłyk , Monika Janeczko , Aleksandra Martyna , Sławomir Czernik , Małgorzata Tokarska-Rodak , et al.
Molecules, 2019, 24 (1), pp.153. ⟨10.3390/molecules24010153⟩
Journal articles hal-02046526v1
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Synthesis of bioactive 2-(arylamino)thiazolo[5,4-f]-quinazolin-9-ones via the Hügershoff reaction or Cu- catalyzed intramolecular C-S bond formation

Damien Hédou , Carole Dubouilh-Benard , N. Loaëc , L. Meijer , Corinne Fruit , et al.
Molecules, 2016, 21 (6), pp.794. ⟨10.3390/molecules21060794⟩
Journal articles hal-02046212v1
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Synthesis of Thiazolo[5,4-f]quinazolin-9(8H)-ones as Multi-Target Directed Ligands of Ser/Thr Kinases

Damien Hédou , Julien Godeau , N. Loaëc , L. Meijer , Corinne Fruit , et al.
Molecules, 2016, 21 (5), pp.578. ⟨10.3390/molecules21050578⟩
Journal articles hal-02046213v1
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6E11, a highly selective inhibitor of Receptor-Interacting Protein Kinase 1, protects cells against cold hypoxia-reoxygenation injury

C. Delehouzé , S. Leverrier-Penna , F. Le Cann , A. Comte , M. Jacquard-Fevai , et al.
Scientific Reports, 2017, 7 (1), pp.12931. ⟨10.1038/s41598-017-12788-4⟩
Journal articles hal-01616456v1
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30th Franco-Belgian conference of pharmacochemistry

Charlotte Bouckaert , Eric Goffin , Sebastien Dilly , Julien Hanson , Lionel Pochet , et al.
Pharmaceuticals, 2016, 9 (4), pp.73. ⟨10.3390/ph9040073⟩
Journal articles hal-02141338v1
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Design, biological evaluation and X-ray crystallography of nanomolar multifunctional ligands targeting simultaneously acetylcholinesterase and glycogen synthase kinase-3

Killian Oukoloff , Nicolas Coquelle , Manuela Bartolini , Marina Naldi , Rémy Le Guével , et al.
European Journal of Medicinal Chemistry, 2019, 168, pp.58-77. ⟨10.1016/j.ejmech.2018.12.063⟩
Journal articles hal-02055769v1
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Marine Natural Products from New Caledonia—A Review

Sofia-Eléna Motuhi , Mohamed Mehiri , Claude Payri , Stéphane La Barre , Stéphane Bach
Marine drugs, 2016, 14 (3), pp.58. ⟨10.3390/md14030058⟩
Journal articles hal-01292225v1
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From drug screening to target deconvolution: A target-based drug discovery pipeline using Leishmania casein kinase 1 isoform 2 to identify compounds with anti-leishmanial activity

Emilie Durieu , Eric Prina , Olivier Leclercq , Nassima Oumata , Nicolas Gaboriaud-Kolar , et al.
Antimicrobial Agents and Chemotherapy, 2016, ⟨10.1128/AAC.00021-16⟩
Journal articles hal-01299756v1
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2-Aminophenones, a common precursor to N-aryl isatins and acridines endowed with bioactivities

Nahida Mokhtari Brikci-Nigassa , Ghenia Bentabed-Ababsa , William Erb , Floris Chevallier , Laurent Picot , et al.
Tetrahedron, 2018, 74 (15), pp.1785-1801. ⟨10.1016/j.tet.2018.02.038⟩
Journal articles hal-01774406v1
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Bioactive Metabolites from the Deep Subseafloor Fungus Oidiodendron griseum UBOCC-A-114129

Marion Navarri , C. Jégou , Arnaud Bondon , Sandrine Pottier , Stéphane Bach , et al.
Marine drugs, 2017, 15 (4), ⟨10.3390/md15040111⟩
Journal articles hal-01518044v1
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Advances in tetrahydropyrido[1,2-a]isoindolone (valmerins) series: Potent glycogen synthase kinase 3 and cyclin dependent kinase 5 inhibitors.

Rajâa Boulahjar , Aziz Ouach , Stéphane Bourg , Pascal Bonnet , Olivier Lozach , et al.
European Journal of Medicinal Chemistry, 2015, 101, pp.274-287. ⟨10.1016/j.ejmech.2015.06.046⟩
Journal articles hal-01212495v1
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Assigning mitochondrial localization of dual localized proteins using a yeast Bi-Genomic Mitochondrial-Split-GFP

Gaétan Bader , Ludovic Enkler , Yuhei Araiso , Marine Hemmerle , Krystyna Binko , et al.
Journal articles hal-02898815v1
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Diversification, Evolution and Sub-Functionalization of 70kDa Heat-Shock Proteins in Two Sister Species of Antarctic Krill: Differences in Thermal Habitats, Responses and Implications under Climate Change

Kévin Cascella , Didier Jollivet , Claire Papot , Nelly Léger , Erwan Corre , et al.
PLoS ONE, 2015, 10 (4), pp.e0121642. ⟨10.1371/journal.pone.0121642⟩
Journal articles hal-01142647v1
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Biological Evaluation of Arylsemicarbazone Derivatives as Potential Anticancer Agents

Anne Cecília Nascimento da Cruz , Dalci José Brondani , Temístocles Ítalo de Santana , Lucas Oliveira da Silva , Elizabeth Fernanda da Oliveira Borba , et al.
Pharmaceuticals, 2019, 12 (4), pp.169. ⟨10.3390/ph12040169⟩
Journal articles hal-03864455v1
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Fused Systems Based on 2-Aminopyrimidines: Synthesis Combining Deprotolithiation-in situ Zincation with N -Arylation Reactions and Biological Properties

Madani Hedidi , Julien Maillard , William Erb , Frédéric Lassagne , Yury S Halauko , et al.
European Journal of Organic Chemistry, 2017, 2017 (39), pp.5903-5915. ⟨10.1002/ejoc.201701004⟩
Journal articles hal-01624382v1
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Screening for Protein-Protein Interaction Inhibitors Using a Bioluminescence Resonance Energy Transfer (BRET)–Based Assay in Yeast

Caroline Corbel , Sara Sartini , Elisabetta Levati , Pierre Colas , Laurent Maillet , et al.
Slas Discovery, 2017, 22 (6), pp.751 - 759. ⟨10.1177/2472555216689530⟩
Journal articles hal-03839336v1
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A combined experimental and theoretical study of the thermal [3+2] cycloaddition of carbonyl ylides with activated alkenes

Samira Hamza-Reguig , Ghenia Bentabed-Ababsa , Luis R Domingo , Mar Ríos-Gutiérrez , Stephanie Philippot , et al.
Journal of Molecular Structure, 2018, 1157, pp.276-287. ⟨10.1016/j.molstruc.2017.12.052⟩
Journal articles hal-01695551v2
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Microalgal biomass of industrial interest: methods of characterization

Catherine Dupré , Hugh D. Burrows , Maria G. Maria G. Campos , Cédric Delattre , Telma Encarnação , et al.
Ange Nzihou. Handbook on Characterization of Biomass, Biowaste and Related By-products, Springer, Heidelberg, pp.537-639, 2020, 978-3-030-35019-2. ⟨10.1007/978-3-030-35020-8_4⟩
Book sections hal-02547368v1