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Synthetic Development of New 3-(4-Arylmethylamino)butyl-5-arylidene-rhodanines under Microwave Irradiation and Their Effects on Tumor Cell Lines and against Protein Kinases
Camille Déliko Dago
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Christelle Ambeu
,
Wacothon-Karime Coulibaly
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Yves-Alain Békro
,
Janat Mamyrbékova
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et al.
Journal articles
hal-01187427v1
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Marine-Derived 2-Aminoimidazolone Alkaloids. Leucettamine B-Related Polyandrocarpamines Inhibit Mammalian and Protozoan DYRK & CLK Kinases
Nadège Loaëc
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Eletta Attanasio
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Benoît Villiers
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Emilie Durieu
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Tania Tahtouh
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et al.
Journal articles
hal-01640115v1
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From Quinoxaline, Pyrido[2,3-b]pyrazine and Pyrido[3,4-b]pyrazine to Pyrazino-Fused Carbazoles and Carbolines
Frédéric Lassagne
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Timothy Langlais
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Elsa Caytan
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Emmanuelle Limanton
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Ludovic Paquin
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et al.
Journal articles
hal-03867783v1
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Synthesis of N-pyridyl azoles using a deprotometalation-iodolysis-N-arylation sequence and evaluation of their antiproliferative activity in melanoma cells
M. Hedidi
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W. Erb
,
G. Bentabed-Ababsa
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Floris Chevallier
,
L. Picot
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et al.
Journal articles
hal-01381138v1
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High-Throughput Screening of marine resources
Arnaud Hochard
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Luc Reininger
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Sandrine Ruchaud
,
Stéphane Bach
Book sections
hal-03871307v1
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Redescription and phylogenetic analyses of Durchoniella spp. (Ciliophora, Astomatida) associated with the polychaete Cirriformia tentaculata (Montagu, 1808)
Laure Sauvadet
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Denis H. Lynn
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Erwan Roussel
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Sophie Le Panse
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Estelle Bigeard
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et al.
Journal articles
hal-01578167v1
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Structure-based design of novel quinoxaline-2-carboxylic acids and analogues as Pim-1 inhibitors
Bruno Oyallon
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Marie Brachet-Botineau
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Cédric Logé
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Pascal Bonnet
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Mohamed Souab
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et al.
Journal articles
hal-03408667v1
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The Anti-Candida albicans Agent 4-AN Inhibits Multiple Protein Kinases
Maciej Masłyk
,
Monika Janeczko
,
Aleksandra Martyna
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Sławomir Czernik
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Małgorzata Tokarska-Rodak
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et al.
Journal articles
hal-02046526v1
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Synthesis of bioactive 2-(arylamino)thiazolo[5,4-f]-quinazolin-9-ones via the Hügershoff reaction or Cu- catalyzed intramolecular C-S bond formation
Damien Hédou
,
Carole Dubouilh-Benard
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N. Loaëc
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L. Meijer
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Corinne Fruit
,
et al.
Journal articles
hal-02046212v1
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Synthesis of Thiazolo[5,4-f]quinazolin-9(8H)-ones as Multi-Target Directed Ligands of Ser/Thr Kinases
Damien Hédou
,
Julien Godeau
,
N. Loaëc
,
L. Meijer
,
Corinne Fruit
,
et al.
Journal articles
hal-02046213v1
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6E11, a highly selective inhibitor of Receptor-Interacting Protein Kinase 1, protects cells against cold hypoxia-reoxygenation injury
C. Delehouzé
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S. Leverrier-Penna
,
F. Le Cann
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A. Comte
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M. Jacquard-Fevai
,
et al.
Journal articles
hal-01616456v1
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30th Franco-Belgian conference of pharmacochemistry
Charlotte Bouckaert
,
Eric Goffin
,
Sebastien Dilly
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Julien Hanson
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Lionel Pochet
,
et al.
Journal articles
hal-02141338v1
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Design, biological evaluation and X-ray crystallography of nanomolar multifunctional ligands targeting simultaneously acetylcholinesterase and glycogen synthase kinase-3
Killian Oukoloff
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Nicolas Coquelle
,
Manuela Bartolini
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Marina Naldi
,
Rémy Le Guével
,
et al.
Journal articles
hal-02055769v1
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Marine Natural Products from New Caledonia—A Review
Sofia-Eléna Motuhi
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Mohamed Mehiri
,
Claude Payri
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Stéphane La Barre
,
Stéphane Bach
Journal articles
hal-01292225v1
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From drug screening to target deconvolution: A target-based drug discovery pipeline using Leishmania casein kinase 1 isoform 2 to identify compounds with anti-leishmanial activity
Emilie Durieu
,
Eric Prina
,
Olivier Leclercq
,
Nassima Oumata
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Nicolas Gaboriaud-Kolar
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et al.
Journal articles
hal-01299756v1
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2-Aminophenones, a common precursor to N-aryl isatins and acridines endowed with bioactivities
Nahida Mokhtari Brikci-Nigassa
,
Ghenia Bentabed-Ababsa
,
William Erb
,
Floris Chevallier
,
Laurent Picot
,
et al.
Journal articles
hal-01774406v1
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Bioactive Metabolites from the Deep Subseafloor Fungus Oidiodendron griseum UBOCC-A-114129
Marion Navarri
,
C. Jégou
,
Arnaud Bondon
,
Sandrine Pottier
,
Stéphane Bach
,
et al.
Journal articles
hal-01518044v1
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Advances in tetrahydropyrido[1,2-a]isoindolone (valmerins) series: Potent glycogen synthase kinase 3 and cyclin dependent kinase 5 inhibitors.
Rajâa Boulahjar
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Aziz Ouach
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Stéphane Bourg
,
Pascal Bonnet
,
Olivier Lozach
,
et al.
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hal-01212495v1
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Assigning mitochondrial localization of dual localized proteins using a yeast Bi-Genomic Mitochondrial-Split-GFP
Gaétan Bader
,
Ludovic Enkler
,
Yuhei Araiso
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Marine Hemmerle
,
Krystyna Binko
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et al.
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hal-02898815v1
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Diversification, Evolution and Sub-Functionalization of 70kDa Heat-Shock Proteins in Two Sister Species of Antarctic Krill: Differences in Thermal Habitats, Responses and Implications under Climate Change
Kévin Cascella
,
Didier Jollivet
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Claire Papot
,
Nelly Léger
,
Erwan Corre
,
et al.
Journal articles
hal-01142647v1
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Biological Evaluation of Arylsemicarbazone Derivatives as Potential Anticancer Agents
Anne Cecília Nascimento da Cruz
,
Dalci José Brondani
,
Temístocles Ítalo de Santana
,
Lucas Oliveira da Silva
,
Elizabeth Fernanda da Oliveira Borba
,
et al.
Journal articles
hal-03864455v1
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Fused Systems Based on 2-Aminopyrimidines: Synthesis Combining Deprotolithiation-in situ Zincation with N -Arylation Reactions and Biological Properties
Madani Hedidi
,
Julien Maillard
,
William Erb
,
Frédéric Lassagne
,
Yury S Halauko
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et al.
Journal articles
hal-01624382v1
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Screening for Protein-Protein Interaction Inhibitors Using a Bioluminescence Resonance Energy Transfer (BRET)–Based Assay in Yeast
Caroline Corbel
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Sara Sartini
,
Elisabetta Levati
,
Pierre Colas
,
Laurent Maillet
,
et al.
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hal-03839336v1
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A combined experimental and theoretical study of the thermal [3+2] cycloaddition of carbonyl ylides with activated alkenes
Samira Hamza-Reguig
,
Ghenia Bentabed-Ababsa
,
Luis R Domingo
,
Mar Ríos-Gutiérrez
,
Stephanie Philippot
,
et al.
Journal articles
hal-01695551v2
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Microalgal biomass of industrial interest: methods of characterization
Catherine Dupré
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Hugh D. Burrows
,
Maria G. Maria G. Campos
,
Cédric Delattre
,
Telma Encarnação
,
et al.
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hal-02547368v1
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