Utilisation de la levure en tant que modèle et outil : de la compréhension de la cytokinèse à l'étude de sélectivité d'une molécule à potentiel thérapeutique
Damien Guiffant
Biologie moléculaire. Rennes 1, 2008. Français.
⟨NNT : ⟩
Theses
tel-01112966v1
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Impact of meriolins, a new class of cyclin-dependent kinase inhibitors, on malignant glioma proliferation and neo-angiogenesis.
Marie Jarry
,
Céline Lecointre
,
Céline Malleval
,
Laurence Desrues
,
Marie-Thérèse Schouft
,
et al.
Neuro-Oncology , 2014, 16 (11), pp.1484-98
Journal articles
hal-01109355v1
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The Anti-Candida albicans Agent 4-AN Inhibits Multiple Protein Kinases
Maciej Masłyk
,
Monika Janeczko
,
Aleksandra Martyna
,
Sławomir Czernik
,
Małgorzata Tokarska-Rodak
,
et al.
Journal articles
hal-02046526v1
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The Plasmodium falciparum, Nima-related kinase Pfnek-4: a marker for asexual parasites committed to sexual differentiation.
Luc Reininger
,
Miguel Garcia
,
Andrew Tomlins
,
Sylke Müller
,
Christian Doerig
Journal articles
inserm-00739795v1
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Synthesis of N-pyridyl azoles using a deprotometalation-iodolysis-N-arylation sequence and evaluation of their antiproliferative activity in melanoma cells
Madani Hedidi
,
Julien Maillard
,
William Erb
,
Frédéric Lassagne
,
Yury Halauko
,
et al.
Journal articles
hal-03875302v1
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High-Throughput Screening of marine resources
Arnaud Hochard
,
Luc Reininger
,
Sandrine Ruchaud
,
Stéphane Bach
Book sections
hal-03871307v1
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Redescription and phylogenetic analyses of Durchoniella spp. (Ciliophora, Astomatida) associated with the polychaete Cirriformia tentaculata (Montagu, 1808)
Laure Sauvadet
,
Denis H. Lynn
,
Erwan Roussel
,
Sophie Le Panse
,
Estelle Bigeard
,
et al.
Journal articles
hal-01578167v1
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Structure-based design of novel quinoxaline-2-carboxylic acids and analogues as Pim-1 inhibitors
Bruno Oyallon
,
Marie Brachet-Botineau
,
Cédric Logé
,
Pascal Bonnet
,
Mohamed Souab
,
et al.
Journal articles
hal-03408667v1
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Synthetic Development of New 3-(4-Arylmethylamino)butyl-5-arylidene-rhodanines under Microwave Irradiation and Their Effects on Tumor Cell Lines and against Protein Kinases
Camille Déliko Dago
,
Christelle Ambeu
,
Wacothon-Karime Coulibaly
,
Yves-Alain Békro
,
Janat Mamyrbékova
,
et al.
Journal articles
hal-01187427v1
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Transcriptome and Peptidome Characterisation of the Main Neuropeptides and Peptidic Hormones of a Euphausiid: The Ice Krill, Euphausia crystallorophias
Jean-Yves Toullec
,
Erwan Corre
,
Benoit Bernay
,
Michael A. S. Thorne
,
Kévin Cascella
,
et al.
Journal articles
hal-01250917v1
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Approches moléculaires de la diversité microbienne de deux environnements extrêmes : les sources hydrothermales profondes et les réservoirs pétroliers
Erwan Corre
Biologie moléculaire. Université de Bretagne Occidentale, 2000. Français.
⟨NNT : ⟩
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tel-01115381v1
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A Haploid System of Sex Determination in the Brown Alga Ectocarpus sp.
Sophia S. Ahmed
,
J. Mark Cock
,
Eugenie Pessia
,
Remy Luthringer
,
Alexandre Cormier
,
et al.
Journal articles
hal-01132642v1
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Sibiriline, a new small chemical inhibitor of receptor-interacting protein kinase 1, prevents immune-dependent hepatitis
F. Le Cann
,
C. Delehouzé
,
S. Leverrier-Penna
,
A. Filliol
,
A. Comte
,
et al.
Journal articles
hal-01616420v1
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Identification de cibles intracellulaires de molécules à activité antiprion
Déborah Tribouillard-Tanvier
Biologie moléculaire. Rennes 1, 2007. Français.
⟨NNT : ⟩
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tel-01118256v1
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Développement de nouveaux inhibiteurs de TgCDPK1 à visée anti-toxoplasmique
Espérance Moine
,
Isabelle Dimier-Poisson
,
Cécile Enguehard-Gueiffier
,
Cedric Logé
,
Mélanie Pénichon
,
et al.
6. Journées du Consortium antiParasitaire et antiFongique : CaPF-2016 " A la croisée des Mondes !" , Consortium Anti-Parasitaire et Fongique (CaPF). FRA., Mar 2016, Tours, France. 49 p
Conference papers
hal-02739722v1
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A yeast-based assay to isolate drugs active against mammalian prions
Stéphane Bach
,
Déborah Tribouillard
,
Nicolas Talarek
,
Nathalie Desban
,
Marc Blondel
Journal articles
hal-02134947v1
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Protein Folding Activity of Ribosomal RNA Is a Selective Target of Two Unrelated Antiprion Drugs
Déborah Tribouillard-Tanvier
,
Suzana dos Reis
,
Fabienne Gug
,
Cécile Voisset
,
Vincent Béringue
,
et al.
Journal articles
hal-02134950v1
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Bioactive Metabolites from the Deep Subseafloor Fungus Oidiodendron griseum UBOCC-A-114129
Marion Navarri
,
C. Jégou
,
Arnaud Bondon
,
Sandrine Pottier
,
Stéphane Bach
,
et al.
Journal articles
hal-01518044v1
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Advances in tetrahydropyrido[1,2-a]isoindolone (valmerins) series: Potent glycogen synthase kinase 3 and cyclin dependent kinase 5 inhibitors.
Rajâa Boulahjar
,
Aziz Ouach
,
Stéphane Bourg
,
Pascal Bonnet
,
Olivier Lozach
,
et al.
Journal articles
hal-01212495v1
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Synthesis of new pyridazino[4,5-b]indol-4-ones and pyridazin-3(2H)-one analogs as DYRK1A inhibitors
Amélie Bruel
,
Romain Bénéteau
,
Mylène Chabanne
,
Olivier Lozach
,
Rémy Le Guevel
,
et al.
Journal articles
hal-01086026v1
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Assigning mitochondrial localization of dual localized proteins using a yeast Bi-Genomic Mitochondrial-Split-GFP
Gaétan Bader
,
Ludovic Enkler
,
Yuhei Araiso
,
Marine Hemmerle
,
Krystyna Binko
,
et al.
Journal articles
hal-02898815v1
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Synthesis and evaluation of the antiproliferative activity of novel thiazoloquinazolinone kinases inhibitors.
Alexandra Testard
,
Laurent Picot
,
Olivier Lozach
,
Melina Blairvacq
,
Laurent Meijer
,
et al.
Journal articles
hal-01443570v1
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Etude de la régulation de deux protéines kinases : GSK-3 et polo
Aline Primot
Biologie cellulaire. Rennes 1, 2001. Français.
⟨NNT : ⟩
Theses
tel-01117984v1
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Synthesis of New N,N'-Bis(5-arylidene-4-oxo-4,5-dihydrothiazolin-2-yl)piperazine Derivatives Under Microwave Irradiation and Preliminary Biological Evaluation.
Wacothon Karime Coulibaly
,
Ludovic Paquin
,
Anoubilé Bénié
,
Yves-Alain Bekro
,
Emilie Durieux
,
et al.
Journal articles
inserm-00864810v1
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Mécanismes d'action des inhibiteurs de kinases cyclines-dépendantes : identification de leurs cibles intracellulaires par chromatographie d'affinité
Marie Knockaert
Biochimie, Biologie Moléculaire. Université de Bretagne Occidentale, 2002. Français.
⟨NNT : ⟩
Theses
tel-01116136v1
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Synthesis, antileishmanial activity and cytotoxicity of 2,3-diaryl- and 2,3,8-trisubstituted imidazo[1,2-a]pyrazines
Pascal Marchand
,
Marc-Antoine Bazin
,
Fabrice Pagniez
,
Guillaume Rivière
,
Lizeth Bodero
,
et al.
Journal articles
hal-03216056v1
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From Peptide Aptamers to Inhibitors of FUR, Bacterial Transcriptional Regulator of Iron Homeostasis and Virulence
Sophie Mathieu
,
Cheickna Cissé
,
Sylvie Vitale
,
Aynur Ahmadova
,
Mélissa Degardin
,
et al.
Journal articles
hal-01354302v1
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Biological Evaluation of Arylsemicarbazone Derivatives as Potential Anticancer Agents
Anne Cecília Nascimento da Cruz
,
Dalci José Brondani
,
Temístocles Ítalo de Santana
,
Lucas Oliveira da Silva
,
Elizabeth Fernanda da Oliveira Borba
,
et al.
Journal articles
hal-03864455v1
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Novel optimization of valmerins (tetrahydropyrido[1,2-a]isoindolones) as potent dual CDK5/GSK3 inhibitors
Aziz Ouach
,
Rajâa Boulahjar
,
Christine Vala
,
Stéphane Bourg
,
Pascal Bonnet
,
et al.
Journal articles
hal-01295635v1
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Conjugating effects of symbionts and environmental factors on gene expression in deep-sea hydrothermal vent mussels.
Isabelle Boutet
,
Raymond Ripp
,
Odile Lecompte
,
Carole Dossat
,
Erwan Corre
,
et al.
Journal articles
inserm-00642454v1
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