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cdc-like/dual-specificity tyrosine phosphorylation-regulated kinases inhibitor leucettine L41 induces mTOR-dependent autophagy: implication for Alzheimer's disease.
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Marine-Derived 2-Aminoimidazolone Alkaloids. Leucettamine B-Related Polyandrocarpamines Inhibit Mammalian and Protozoan DYRK & CLK Kinases
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Synthesis and biological evaluation of tetrahydro[1,4]diazepino[1,2-a]indol-1-ones as cyclin-dependent kinase inhibitors
Putey Aurelien
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From Quinoxaline, Pyrido[2,3-b]pyrazine and Pyrido[3,4-b]pyrazine to Pyrazino-Fused Carbazoles and Carbolines
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Structure-based design of novel quinoxaline-2-carboxylic acids and analogues as Pim-1 inhibitors
Bruno Oyallon
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Synthesis of N-pyridyl azoles using a deprotometalation-iodolysis-N-arylation sequence and evaluation of their antiproliferative activity in melanoma cells
M. Hedidi
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Microwave synthesis of new 3-(3-aminopropyl)-5-arylidene-2-thioxo-1,3-thiazolidine-4-ones as potential Ser/Thr protein kinase inhibitors
Camille Déliko Dago
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Synthesis of N-pyridyl azoles using a deprotometalation-iodolysis-N-arylation sequence and evaluation of their antiproliferative activity in melanoma cells
Madani Hedidi
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Acridone Alkaloids from Glycosmis chlorosperma as DYRK1A Inhibitors
Mehdi A. Beniddir
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Erell Le Borgne
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Development of new highly potent imidazo[1,2-b]pyridazines targeting Toxoplasma gondii calcium-dependent protein kinase 1
Espérance Moine
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Isabelle Dimier-Poisson
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The Anti-Candida albicans Agent 4-AN Inhibits Multiple Protein Kinases
Maciej Masłyk
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Monika Janeczko
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hal-02046526v1
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Synthesis of bioactive 2-(arylamino)thiazolo[5,4-f]-quinazolin-9-ones via the Hügershoff reaction or Cu- catalyzed intramolecular C-S bond formation
Damien Hédou
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hal-02046212v1
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Synthesis of Thiazolo[5,4-f]quinazolin-9(8H)-ones as Multi-Target Directed Ligands of Ser/Thr Kinases
Damien Hédou
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Corinne Fruit
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hal-02046213v1
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6E11, a highly selective inhibitor of Receptor-Interacting Protein Kinase 1, protects cells against cold hypoxia-reoxygenation injury
C. Delehouzé
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hal-01616456v1
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30th Franco-Belgian conference of pharmacochemistry
Charlotte Bouckaert
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Eric Goffin
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Sebastien Dilly
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Julien Hanson
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Design, biological evaluation and X-ray crystallography of nanomolar multifunctional ligands targeting simultaneously acetylcholinesterase and glycogen synthase kinase-3
Killian Oukoloff
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Nicolas Coquelle
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Manuela Bartolini
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Rémy Le Guével
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hal-02055769v1
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From drug screening to target deconvolution: A target-based drug discovery pipeline using Leishmania casein kinase 1 isoform 2 to identify compounds with anti-leishmanial activity
Emilie Durieu
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hal-01299756v1
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2-Aminophenones, a common precursor to N-aryl isatins and acridines endowed with bioactivities
Nahida Mokhtari Brikci-Nigassa
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Ghenia Bentabed-Ababsa
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Further investigation of Paprotrain: Towards the conception of selective and multi-targeted CNS kinase inhibitors
Christophe Labrière
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Olivier Lozach
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Mélina Blairvacq
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Laurent Meijer
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Catherine Guillou
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Bioactive Metabolites from the Deep Subseafloor Fungus Oidiodendron griseum UBOCC-A-114129
Marion Navarri
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C. Jégou
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Advances in tetrahydropyrido[1,2-a]isoindolone (valmerins) series: Potent glycogen synthase kinase 3 and cyclin dependent kinase 5 inhibitors.
Rajâa Boulahjar
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Aziz Ouach
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Stéphane Bourg
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Pascal Bonnet
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Olivier Lozach
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Biological Evaluation of Arylsemicarbazone Derivatives as Potential Anticancer Agents
Anne Cecília Nascimento da Cruz
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Dalci José Brondani
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Temístocles Ítalo de Santana
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Lucas Oliveira da Silva
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Elizabeth Fernanda da Oliveira Borba
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hal-03864455v1
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New 5-ylidene rhodanine derivatives based on the dispacamide A model.
Solène Guihéneuf
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Ludovic Paquin
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François Carreaux
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Fused Systems Based on 2-Aminopyrimidines: Synthesis Combining Deprotolithiation-in situ Zincation with N -Arylation Reactions and Biological Properties
Madani Hedidi
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Julien Maillard
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William Erb
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Frédéric Lassagne
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Yury S Halauko
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hal-01624382v1
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Synthesis and molecular modelling studies of 8-arylpyrido[3',2':4,5thieno[3,2-d]pyrimidin-4-amines as multitarget Ser/Thr kinases inhibitors
Yvonnick Loidreau
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Emmanuel Deau
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Pascal Marchand
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Marie-Renée Nourrisson
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Cédric Logé
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hal-01135195v1
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A combined experimental and theoretical study of the thermal [3+2] cycloaddition of carbonyl ylides with activated alkenes
Samira Hamza-Reguig
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Ghenia Bentabed-Ababsa
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Luis R Domingo
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Mar Ríos-Gutiérrez
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Stephanie Philippot
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hal-01695551v2
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Tampering with Cell Division by Using Small-Molecule Inhibitors of CDK-CKS Protein Interactions
Amel Hamdi
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Aurélien Lesnard
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Peggy Suzanne
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Thomas Robert
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Maria A. Miteva
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istex
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